Trestolone (7alpha-methyl-19-n/testosterone/ Ment)or trestolone was one of several 19-nortestosterone derivatives considered a possible male contraceptive therapy due to its unique chemical properties. Initially, pharmaceutical companies combined progesterone with testosterone to produce a viable male contraceptive option due to progesterone’s ability to suppress spermatogenesis.
Trestolone is unable to bind to 5alpha-reductase and therefore cannot convert to DHT, making it a perfect candidate for an androgenic male contraceptive.
Theoretically, trestolone has a ratio of 2300-650, which means it is 23 times more anabolic than testosterone and 6.5 times more androgenic. But a 1992 study in rats found that the anabolic potency of this drug is 10 times greater than that of testosterone, while being 12 times more suppressive on HTPA.
The reason for this lies in the unique alpha-methyl group on carbon 7 of the molecule. This methyl group protrudes beneath the steroid ring structure and sterically inhibits the conversion to DHT. However, Trestolone can still undergo aromatization and undergo other androgen-dependent functions, making it act effectively like testosterone in the body despite being a derivative of 19-nortestosterone.
Trestolone has also been shown to have minimal affinity for progesterone and mineralocorticoid receptors, despite being a derivative of nandrolone.
Testosterone is an anabolic steroid that initiates a fairly strong increase in muscle mass, which also significantly increases the dynamics of the protein synthesis process in the body.
Minors should not use this drug because it can cause an unnatural and greatly accelerated sexual maturation process.
Trestolone was initially created mainly to create an androgen replacement, this synthetic (or artificial) steroid was used, which is considered quite powerful.
Purposes of medical use of trestolone include, among others: a contraceptive session, rapid bone loss, benign prostatic hyperplasia, prostate cancer, primary hypogonadism, cachexia (a disease involving the so-called muscle wasting syndrome), sarcopenia , induced anabolism, and typically male alopecia.
EFFECTS:
Extremely anabolic compound 10 to 23 times higher than testosterone.
It is extremely powerful in helping users destroy fat & Build muscle.
Increased strength and muscle mass.
Does not bind to SHBG.
Does not convert to DHT.
No significant increase in hematocrit or hemoglobin.
Quick effect.
High appetite.
SIDE EFFECTS:
Significant increase in systolic blood pressure.
Rapid estrogen conversion.
Dry throat.
Excessive sweating.
Stomach upset.
Diarrhea.
Heartburn.
Back acne.
Insomnia.
Night sweats.
Fluctuations in our mood.
It is strongly recommended that you use an aromatase inhibitor such as Arimidex or Letrozole while taking Trestolone.
Appetite should be extremely high and you should see a slight increase in strength in the gym. 1.25 mg letrozole every other day to combat conversion to 7a-methyl estradiol.
DOSAGE:
Beginner: 100 mg per week.
Intermediate: 200 mg per week.
Advanced: 300 mg per week.
It is recommended to start by taking 100 mg of Trestolone acetate per week, to see how your body responds. If your body responds well, you may consider slowly increasing the dosage, up to 300 mg per week.
Reviews
There are no reviews yet.